 Bradykinin Receptor Antagonists
"Bradykinin Receptor Antagonists" is a descriptor in the National Library of Medicine's controlled vocabulary thesaurus,
MeSH (Medical Subject Headings). Descriptors are arranged in a hierarchical structure,
which enables searching at various levels of specificity.
Compounds and drugs that inhibit ligand binding or cellular signaling by BRADYKININ RECEPTORS.
| Descriptor ID |
D065168
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| MeSH Number(s) |
D27.505.519.265
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| Concept/Terms |
Bradykinin Receptor Antagonists- Bradykinin Receptor Antagonists
- Antagonists, Bradykinin Receptor
- Receptor Antagonists, Bradykinin
- Bradykinin Receptor Blockers
- Receptor Blockers, Bradykinin
- Bradykinin Receptor Inhibitors
- Inhibitors, Bradykinin Receptor
- Receptor Inhibitors, Bradykinin
- Bradykinin Antagonists
- Antagonists, Bradykinin
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Below are MeSH descriptors whose meaning is more general than "Bradykinin Receptor Antagonists".
Below are MeSH descriptors whose meaning is more specific than "Bradykinin Receptor Antagonists".
This graph shows the total number of publications written about "Bradykinin Receptor Antagonists" by people in this website by year, and whether "Bradykinin Receptor Antagonists" was a major or minor topic of these publications.
To see the data from this visualization as text, click here.
| Year | Major Topic | Minor Topic | Total |
|---|
| 2002 | 3 | 0 | 3 | | 2014 | 0 | 1 | 1 |
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Below are the most recent publications written about "Bradykinin Receptor Antagonists" by people in Profiles.
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Chen Y, Gera L, Zhang S, Li X, Yang Y, Mamouni K, Wu AY, Liu H, Kucuk O, Wu D. Small molecule BKM1972 inhibits human prostate cancer growth and overcomes docetaxel resistance in intraosseous models. Cancer Lett. 2019 04 01; 446:62-72.
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Malbr?n A, Riedl M, Ritchie B, Smith WB, Yang W, Banerji A, H?bert J, Gleich GJ, Hurewitz D, Jacobson KW, Bernstein JA, Khan DA, Kirkpatrick CH, Resnick D, Li H, Fern?ndez Romero DS, Lumry W. Repeat treatment of acute hereditary angioedema attacks with open-label icatibant in the FAST-1 trial. Clin Exp Immunol. 2014 Aug; 177(2):544-53.
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Gera L, Roy C, Bawolak MT, Charest-Morin X, Marceau F. N-terminal extended conjugates of the agonists and antagonists of both bradykinin receptor subtypes: structure-activity relationship, cell imaging using ligands conjugated with fluorophores and prospect for functionally active cargoes. Peptides. 2012 Apr; 34(2):433-46.
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Stewart JM, Chan DC, Simkeviciene V, Bunn PA, Helfrich B, York EJ, Taraseviciene-Stewart L, Bironaite D, Gera L. Bradykinin antagonists as new drugs for prostate cancer. Int Immunopharmacol. 2002 Dec; 2(13-14):1781-6.
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Chan DC, Gera L, Stewart JM, Helfrich B, Zhao TL, Feng WY, Chan KK, Covey JM, Bunn PA. Bradykinin antagonist dimer, CU201, inhibits the growth of human lung cancer cell lines in vitro and in vivo and produces synergistic growth inhibition in combination with other antitumor agents. Clin Cancer Res. 2002 May; 8(5):1280-7.
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Taraseviciene-Stewart L, Gera L, Hirth P, Voelkel NF, Tuder RM, Stewart JM. A bradykinin antagonist and a caspase inhibitor prevent severe pulmonary hypertension in a rat model. Can J Physiol Pharmacol. 2002 Apr; 80(4):269-74.
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Banik RK, Kozaki Y, Sato J, Gera L, Mizumura K. B2 receptor-mediated enhanced bradykinin sensitivity of rat cutaneous C-fiber nociceptors during persistent inflammation. J Neurophysiol. 2001 Dec; 86(6):2727-35.
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Larriv?e JF, Gera L, Houle S, Bouthillier J, Bachvarov DR, Stewart JM, Marceau F. Non-competitive pharmacological antagonism at the rabbit B(1) receptor. Br J Pharmacol. 2000 Nov; 131(5):885-92.
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Reissmann S, Pineda F, Vietinghoff G, Werner H, Gera L, Stewart JM, Paegelow I. Structure activity relationships for bradykinin antagonists on the inhibition of cytokine release and the release of histamine. Peptides. 2000 Apr; 21(4):527-33.
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Sejbal J, Wang Y, Cann JR, Stewart JM, Gera L, Kotovych G. A comparative NMR and molecular dynamics study of the conformations of bradykinin B1 and B2, B2, and B1-specific receptor antagonists B-9430, B-9436, and B-9858. Biopolymers. 1997 Oct 15; 42(5):521-35.
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